富山県立大学工学部 医薬品工学科 バイオ医薬品工学講座

安田研究室

                                                      

2021

2021年

  1. Elucidation of metabolic pathways of 25-hydroxyvitamin D3 mediated by CYP24A1 and CYP3A using Cyp24a1 knockout rats generated by CRISPR/Cas9 system
    Yasuda K, Nishikawa M, Okamoto K, Horibe K, Mano H, Yamaguchi M, Nakagawa K, Tsugawa N, Okano T, Kawagoe F, Kittaka A, Ikushiro S, Sakaki T.
    J. Biol. Chem., in press (2021)


  2. Chemical Synthesis of Side-Chain-Hydroxylated Vitamin D3 Derivatives and Their Metabolism by CYP27B1.
    Ryota Sakamoto, Akiko Nagata, Haruki Ohshita, Yuka Mizumoto, Miho Iwaki, Kaori Yasuda, Toshiyuki Sakaki, Kazuo Nagasawa
    Chembiochem : a European journal of chemical biology 22(19) 2896-2900 (2021)


  3. Epicatechin gallate and epigallocatechin gallate are potent inhibitors of human arylacetamide deacetylase.
    Yasuda K, Watanabe K, Fukami T, Nakashima S, Ikushiro S, Nakajima M, Sakaki T.,
    Drug Metab Pharmacokinet., in press (2021)


  4. Development of In Vitro and In Vivo Evaluation Systems for Vitamin D Derivatives and Their Application to Drug Discovery
    Kaori Yasuda, Miyu Nishikawa, Hiroki Mano, Masashi Takano, Atsushi Kittaka, Shinichi Ikushiro,Toshiyuki Sakaki
    International Journal of Molecular Sciences 22(21) 11839-11839 (2021)


  5. Stereoselective Synthesis of 24-Fluoro-25-Hydroxyvitamin D3 Analogues and Their Stability to hCYP24A1-Dependent Catabolism
    Fumihiro Kawagoe, Sayuri Mototani, Kaori Yasuda, Hiroki Mano, Toshiyuki Sakaki, Atsushi Kittaka
    International Journal of Molecular Sciences 22(21) 11863-11863 (2021)


  6. 代謝研究より明らかになりつつあるビタミンD群の生理作用
    西川美宇、安田佳織、生城真一、榊利之;
    バイオサイエンスとインダストリー, 79:12-15 (2021)


メニュー

コンテンツへスキップ
  • トップページ

Copyright ©富山県立大学工学部 医薬品工学科 バイオ医薬品工学講座安田研究室 , All rights reserved.